Company* (Symbol)

Product

Description

Indication

Status (Date)

CANCER

Allos Therapeutics Inc. (ALTH)

RSR13

Synthetic allosteric modifier of hemoglobin that noncovalently binds to hemoglobin, increasing oxygen delivery to hypoxic tissue

Non-small-cell lung cancer

Completed patient enrollment in a Phase II trial in patients undergoing chemotherapy followed by radiation therapy (8/2)

Celgene Corp. (CELG)

Thalomid (FDA- approved)

Thalidomide; thought to act by modulating levels of tumro necrosis factor-alpha

Advanced colorectal cancer

Published interim analysis of a pilot trial combining Thalomid with irinotecan in The Lancet (8/11)

Cell Pathways Inc. (CLPA)

CP461

Compound that triggers selective apoptosis in neo-plastic cells by inhibiting cyclic GMP phosphodiesterase

Cancer

Completed Phase IB testing with encouraging safety results (8/3)

Cel-Sci Corp. (AMEX:CVM)

Multikine

Natural mixture of human cytokines, including interleukin-2

Head and neck cancer

Presented updated Phase I/II findings showing tumor elimin- ation, tumor reduction and activa- tion of the immune system; data were reported at the 5th Interna- tional Congress on Head and Neck Cancer in San Francisco (8/3)

Corixa Corp. (CRXA)

Melacine

Therapeutic cancer vaccine made of lysed cells from 2 melanoma cell lines with a broad array of melanoma antigens, combined with Detox adjuvant (contains monophosphoryl lipid A and mycobacterial cell- wall skeleton)

Stage IV metastatic melanoma

Completed a 253-patient Phase III trial comparing Melacine and Intron A therapy with Intron A alone (8/16)

Inex Pharmaceuticals Corp. (Canada; INEX)

Onco-TCS

Therapeutic consisting of vincristine encapsulated in Inex's transmembrane carrier systems drug delivery technology

Small-cell lung cancer

Initiated Phase II trial (8/23)

Inex Pharmaceuticals Corp. (Canada; INEX)

Onco TCS

Therapeutic consisting of vincristine encapsulated in Inex's transmembrane carrier systems drug delivery technology

Relapsed solid tumors in children and adolescents

Initiated second Phase II trial to broaden development for Onco TCS beyond relapsed aggressive non-Hodgkin's lymphoma (8/24)

Intracel Corp.*

HumaRAD

Fully human monoclonal antibody-based product that delivers radiation directly to a tumor

Head and neck cancer

Demonstrated safety and feasibility in a 10-patient pilot study (8/2)

Intracel Corp.*

OncoVAX

Cancer vaccine; incorporates recombinant prostate-specific antigen plus adjuvant in liposomal formulation

Stage II colon cancer

Reported finding of three trials demonstrating significant improvement in the recurrence- free interval and recurrence-free survival (8/31)

LifeTime Pharmaceuticals*

Beta LT

Beta-alanyl cysteamine disulfide; synthetic small- molecule immune stimulator

Cancer

Announced early closure of both initial Phase I/II trials, which have achieved all targeted goals (8/2)

Ligand Pharmaceuticals Inc. (LGND)

Targretin Capsules (FDA- approved)

Bexarotene; synthetic retinoid analogue that selectively activates retinoid X receptors; oral formulation

Non-small-cell lung cancer

Follow-up study showed Targretin capsules in combination with chemotherapy may increase patient survival (8/14)

Oxigene Inc. (OXGN)

Declopramide

Oral formulation of DNA repair inhibitor based on the N-substituted benzamide class of compounds

Advanced-stage solid tumors

Announced results of two Phase I trials to be presented at the 25th ESMO Congress in Hamburg (8/1)

Pfizer Inc. (NYSE:PFE)

Prinomastat

Matrix metalloprotease inhibitor

Advanced hormone-refractory prostate cancer and advanced non- small-cell lung cancer

Two Phase III clinical trials were halted when the product failed to meet efficacy objectives in combination with standard chemotherapy (8/4)

Scotia Holdings plc (UK; LSE:SOH)

Foscan

Temoporfin, mTHPC; photodynamic therapeutic that uses non-thermal lasers to activate light-sensitive drug

Head and neck cancer

Presented results from trials on more than 250 patients at the 5th International Conference on Head and Neck Cancer in San Francisco (8/2)

SuperGen Inc. (SUPG) and Abbott Laboratories (NYSE:ABT)

Rubitecan

Oral chemotherapy in the camptothecin class

Various cancers

The company said Phase III trials are "continuing full force" despite some delays; the company targets an NDA for mid-2001 (8/31)

Techniclone Corp. (TCLN)

Cotara

Tumor necrosis therapy; chimeric monoclonal anti- body that targets DNA-associated histone antigens, labeled with I-131 (targets necrotic center of tumor)

Brain cancer

Expanded Phase II trial to include Northwestern University (8/3)

Vical Inc. (VICL)

Allovectin-7

DNA/lipid complex containing the human gene encoding the HLA- B7 antigen; intra-tumoral injection

Head and neck cancer

Released results from Phase I and Phase II studies showing Allovectin-7 to be safe (8/1)

Vion Pharmaceuticals Inc. (VION)

TAPET bacterial vector

Tumor amplified protein expression therapy; Salmon- ella vector consisting of highly attenuated bacteria that preferentially replicate in tumors

Advanced cancer

Initiated a Phase I intravenous trial at Beth Israel Deaconess Medical Center; study is expected to enroll 20 to 30 patients (8/25)

Xcyte Therapies Inc.*

Xcellerated T cells

Patient blood is collected and the T cells are stimulated to increase 100- fold and are injected into the patient; process uses anti-CD3 and anti-CD28 monoclonal antibodies covalently attached to superparamagnetic microbeads (designed to mimic antigenpresenting cells); the complexes activate T cells and the microbeads are then removed

Metastasized kidney cancer

Initiated a clinical study in 20 patients at the University of Calif., Los Angeles (8/2)

CARDIOVASCULAR

Aquasearch Inc. (OTCBB:AQSE)

AstaFactor (astaxanthin)

Oral astaxanthin-rich algae extract

Coronary heart disease

Initiated a randomized, double-blind trial evaluating 100 patients (8/22)

Centocor Inc. (subsidiary of Johnson & Johnson [NYSE:JNJ]) and Eli Lilly and Co. (NYSE:LLY)

ReoPro (FDA- approved)

Abciximab; a multirecep tor monoclonal antibody inhibitor of glycoprotein IIb/IIIa (alpha V beta 3) and MAC-1 plasty or bypass)

Unstable angina and non-ST eleva- tion myocardial infarction when a coronary intervention (angioed at 458 sites worldwide; data is not planned

Presented results of a Phase III trial showing ReoPro didn't provide a statistically significant benefit over placebo; the trial was double-blind, randomized and placebo-controlled and conduct from the GUSTO IV ACS (Global Use of Strategies to Open Occluded Arteries in Acute Coronary Syndrome) trial were presented at the 22nd meeting of the European Society of Cardiology in Amsterdam (8/28)

Genentech Inc. (NYSE:DNA)

TNKase (FDA- approved)

Tenecteplase; second-generation, single-bolus recombinant plasminogen activator with greater specificity to fibrin than Genentech's first- generation tissue plasminogen activator (Activase)

Heart attack

Reported one-year follow-up data at the 22nd annual congress of the European Society of Cardiology in Amsterdam; results were from ASSENT II trial (Assessment of the Safety and Efficacy of a New Thrombolytic agent) (8/29)

GenVec Inc.*

BioBypass

Angiogenic gene therapy that delivers vascular endothelial growth factor 121

Peripheral vascular disease

Began a double-blind, placebocontrolled Phase II trial in 100 patients with ischemic leg pain who are not candidates for other procedures (8/10)

Myogen Inc.*

Enoximone

Phosphodiesterase (type III) inhibitor; oral formulation

Heart disease

Published findings that low doses of enoximone improve exercise ability of patients with heart failure in a double-blind, placebo- controlled study; data were published in the Journal of the American College of Cardiology (8/23)

United Therapeutics Corp. (UTHR)

Uniprost

Subcutaneous prostacyclin therapy; stable structural analogue of prostacyclin

Pulmonary hypertension

Presented data from Phase III trial at the 22nd meeting of the European Society of Cardiology in Amsterdam (8/28)

CENTRAL NERVOUS SYSTEM

Guilford Pharmaceuticals Inc. (GLFD) and Amgen Inc. (AMGN)

Neuroimmunophilin ligands

Orally-active drugs shown to cross the blood-brain barrier in order to induce nerve growth

Parkinson's disease

Commenced a Phase II trial to evaluate safety and efficacy; trial is double-blind, randomized and placebo-controlled (8/7)

Repligen Corp. (RGEN)

Secretin

Synthetic porcine secretin

Autism

Presented study results showing changes in the metabolic profiles in autistic children treated with secretin; data were reported at the World Congress of Pediatric Gastroenterology in Boston (8/9)

Sepacor Inc. (SEPR)

(S)-zopiclone

Single-isomer version of zopiclone, a non-benzodiazepine, rapid-acting hypnotic

Insomnia

Completed enrollment in 400 patient efficacy trial; Phase III studies slated to begin in third quarter (8/28)

INFECTION

Amrad Corp. Ltd. (Australia; ASX:AMC)

AM365

Inhibitor of viral replication

Hepatitis B

Completed a Phase I trial showing a specificity for Hepatitis B virus by the drug and selectivity for the virus rather than the host (8/30)

GelTex Pharmaceuticals Inc. (GELX)

GT160-246

Non-antibiotic toxin binding polymer

Clostridium difficile colitis

Completed a double-blind, placebo-controlled, randomized study of three doses in 24 normal Volunteers (8/22)

InterMune Pharmaceuticals Inc. (ITMN)

Actimmune (aerosolized)

Interferon gamma-1b; aerosolized formulation

Pulmonary multidrug- resistant tuberculosis

Commenced enrollment for a Phase III trial evaluating safety and efficacy of aerosolized Actimmune (8/1)

Interneuron Pharmaceuticals Inc. (IPIC)

PRO 2000 Gel

Microbicide designed to provide protection against HIV infection and other sexually transmitted diseases

Prevention of HIV infection and other sexually transmitted diseases

Enrolled the first HIV patients into a government-sponsored Phase I/II safety study (8/17)

OXO Chemie Inc. (subsidiary of OXO Chemie AG; Switzerland)

WF10

Macrophage regulation drug containing proprietary chlorite

Late-stage HIV disease

Completed enrollment in Phase III trial (8/8)

PathoGenesis Corp. (PGNS)

TOBI (FDA- approved)

Tobramycin solution for inhalation

Bronchiectasis

Published study in the American Journal of Respiratory and Critical Care Medicine of a double-blind, placebo-controlled, randomized study of 74 patients (8/24)

PathoGenesis Corp. (PGNS)

TOBI (FDA- approved)

Tobramycin solution for inhalation

Ventilator- associated pneumonia

Initiated enrollment in a Phase I open-label study (8/29)

Triangle Pharmaceuticals Inc. (VIRS)

Coactinon

Emivirine; non-nucleoside reverse transcriptase inhibitor

HIV infection

Company said it would continue development following FDA's 12/99 notification that additional Phase III studies would be required; Triangle plans to enroll an additional 280 patients in the Phase III study, MKC-401, in which Coactinon is being evaluated in combination with d4T (stavudine) and Coviracil (8/10)

Vical Inc. (VICL), Aventis Pasteur (unit of Aventis SA [France; NYSE:AVE]) and the U.S. Navy

MuStDO 5

Multigene vaccine incorporating five genes for Plasmodium falciparum antigens, plus a naked DNA agent encoding granulocyte macrophage colony stimulating factor, an immune stimulant

Prevention of infection with the malaria parasite, Plasmodium falciparum

Initiated a clinical trial to test the safety, immunogenicity and protective efficacy; trial is a Phase II dose-escalation study (8/22)

MISCELLANEOUS

Alza Corp. (NYSE:AZA)

Ditropan XL (FDA- approved)

Once-daily formulation of oxybutinin

Overactive bladder

Cleveland Clinic researchers presented positive clinical data showing the drug improved quality of life with fewer discontinuations due to adverse events than conventional oxybutinin; results were presented at the International Continence Society's 30th annual meeting in Tampere, Finland (8/31)

Alexion Pharmaceuticals Inc. (ALXN)

5G1.1

Monoclonal antibody that inhibits the fifth component of the complement cascade

Rheumatoid arthritis

Completed patient enrollment in a multicenter, double-blind, randomized, placebo-controlled Phase II trial; trial involves 200 patients (8/24)

Angiotech Pharmaceuticals Inc. (ANPI)

Topical Paclitaxel Gel

Yew tree-derived semisynthetic taxoid; inhibits abnormal skin cell growth, inflammatory cell response and angiogenesis

Psoriasis

Announced results of two Phase I trials conducted at Harvard University and the University of British Columbia (8/22)

BioTime Inc. (AMEX:BTX)

PentaLyte

Pentastarch-based physiologically balanced blood plasma volume expander

To expand blood plasma volume

Completed a Phase I trial (8/30)

Idec Pharmaceuticals Corp. (IDPH)

Clenoliximab (IDEC-151)

Primatized, non-depleting, anti-CD4 monoclonal antibody believed to regulate helper T-cell function

Rheumatoid arthritis

Began a multicenter, double- blind, randomized, placebo-controlled study evaluating multiple doses of the agent used in combination with methotrexate (8/7)

Novavax Inc. (AMEX:NOX)

Androsorb

Topical cream formulation containing nanosome- encapsulated testosterone

Testosterone deficiency

Began enrolling post-menopausal women in a Phase I study assessing the safety of Androsorb (8/10)

Symbollon Corp. (SYMBA)

IoGen

Molecular iodine

Fibrocystic breast disease

Company announced preliminary results of a Phase II trial (8/16)

Notes:

* Privately held

Unless otherwise noted, the stock symbols listed for public companies are on the Nasdaq market.

AMEX = American Stock Exchange; CDNX = Canadian Venture Exchange; LSE = London Stock Exchange; NYSE = New York Stock Exchange; OTC BB = Over the Counter Bulletin Board; SSE = Swedish Stock Exchange; TSE = Toronto Stock Exchange

ND = Not disclosed