Company* (Symbol)

Product

Description

Indication

Status (Date)**

CANCER

Calydon Inc.*

CV787

Second-generation virus; a prostate-specific gene incorporated into an attenuated adenovirus

Prostate cancer patients seeking alternatives to radiation or radical surgery

Commenced Phase I/II trial (10/25)

Cell Pathways Inc. (CLPA)

Aptosyn (Exisulind)

A selective apoptotic, anti-neoplastic compound that inhibits a cyclic GMP phosphodiesterase and selectively induces apoptosis in abnormally growing precancerous and cancerous cells, but not in normal cells

Familial adenomatous polyposis

Reported clinical trial data (10/27)

Cell Therapeutics Inc. (CTIC)

Lisofylline

A small-molecule anti-inflammatory compound that works by modulating selective stress-activated cell signaling pathways that respond to chemotherapy, radiation and trauma, reducing oxidative damage to tissues

Acute myeloid leukemia

Reported results of Phase III trial (10/11)

ImClone Systems Inc. (IMCL)

C225

Monoclonal antibody antagonist to the epidermal growth factor receptor, which is associated with the growth and survival of cancer cells in a variety of solid tumors

Refractory colorectal carcinoma

Initiated enrollment in a Phase II trial evaluating C225 in combination with the chemotherapeutic agent CPT-11 (10/8)

The Immune Response Corp. (IMNR)

Patented vaccine technology that uses tumor cells mixed with fibroblasts that are genetically engineered to secrete the IL-2 cytokine in order to stimulate the immune system against tumors

Colon cancer

Reported Phase I results in the September 1999 issue of Clinical Cancer Research (10/11)

Matrix Pharmaceutical Inc. (MATX)

FMdC

Systemically administered nucleoside analogue

Non-small-cell lung cancer

Completed patient enrollment in Phase II trial (10/4)

Neopharm Inc. (AMEX:NEO)

IL13 PE38QQR (IL 13-toxin)

A targeted cytotoxin that uses the IL-13 receptor on the surface of cancer cells to deliver a bacterial toxin (PE38QQR), which has been shown to destroy tumor cells, but not normal cells

Renal cell carcinoma

Initiated Phase I trial (10/18)

OxiGene Inc. (Sweden; OXGN; SSE:OXGN)

Combretastatin A4 Prodrug (CA4P)

Angiogenic inhibitor that attacks pre-existent tumor vasculature

Various cancers

Announced interim results of Phase I trial (10/4)

Procept Inc. (PRCT)

06-Benzylguanine

A chemosensitizer that acts by inactivating tumor AGT, a DNA repair protein that interferes with the effectiveness of 06-alkylating chemotherapeutic agents

Multiple myeloma

Initiated Phase I trial of 06-Benzylguanine in combination with the chemotherapeutic drug carmustine (10/20)

Progenics Pharmaceuticals Inc. (PGNX) and Bristol-Myers Squibb Co. (NYSE:BMY)

GMK vaccine

Vaccine designed to stimulate the immune system to control or eradicate residual cancer cells following tumor removal

Malignant melanoma

Completed patient enrollment in Phase III trial (10/6)

StressGen Biotechnologies Corp. (Canada; TSE:SSB)

HspE7

A recombinant fusion product composed of heat shock protein 65 (Hsp65) from M. Bovis BCG and the protein E7, a tumor specific antigen derived from the human papillomavirus

High-grade anal dysplasia

Commenced Phase I trial (10/25)

Techniclone Corp. (TCLN)

Cotara

Tumor necrosis therapy; chimeric monoclonal antibody that targets DNA-associated histone antigens, labeled with I-131 (targets necrotic center of tumor)

Various solid tumor cancers

Presented Phase I data at the 13th Annual International Congress on Brain Tumor Research in Japan (10/4)

Therion Biologics Corp.* and the National Cancer Institute

Two recombinant fowlpox and vaccinia viral vectors encoding tyrosinase, which has been shown to be commonly expressed in metastatic melanoma tumors; products are in vaccine form

Metastatic melanoma

Initiated Phase II trial of two therapeutic vaccines alone and in combination with interleukin-2 (10/18)

Vical Inc. (VICL)

Leuvectin

Gene-encoding interleukin-2 (complexed with lipid) administered by direct intratumoral injection

Kidney cancer

Reported Phase I/II results in the October issue of the Journal of Clinical Oncology (10/4)

CARDIOVASCULAR

AtheroGenics Inc.*

AGI-1067

Orally deliverable, chemically engineered compound that provides direct vascular protection and reduces high LDL cholesterol levels

Post-angioplasty restenosis

Commenced Phase II trial (10/12)

Cerus Corp. (CERS)

S-303

Pathogen inactivation system that targets and inactivates blood-borne pathogens, while leaving the therapeutic properties of red blood cells intact

Red blood cells intended for transfusion

Reported results of Phase Ib trial (10/26)

Corvas International Inc. (CVAS)

rNAPc2

Injectable anticoagulant recombinant protein, discovered in its original form in blood-feeding hookworms

Patients undergoing percutaneous transluminal coronary angioplasty, and the occurrence of clinically overt bleeding

Commenced a second, multi-center Phase II trial (10/28)

CytRx Corp. (CYTR)

Flocor

Purified poloxamer 188; intravenously delivered surfactant molecule that alters the way cells and molecules interact with water

Acute sickle cell crisis

Completed patient enrollment in Phase III trial

The Medicines Co.* and Duke University Medical Institute

Angiomax (bivalirudin)

An anticoagulant therapeutic that directly inhibits thrombin, a key component in blood clot formation and extension

Patients at risk for heparin-induced thrombocytopenia and heparin-induced thrombocytopenia and thrombosis syndrome during coronary procedures

Initiated an expanded access safety and efficacy study (10/28)

Scios Inc. (SCIO)

Natrecor (nesiritide)

A recombinant form of B-type natriuretic peptide, a naturally occurring hormone that aids healthy functioning of the heart

Vasodilation in the management of acute congestive heart failure

Commenced patient enrollment for a Phase III trial (10/27)

Texas Biotechnology Corp. (AMEX:TXB)

TBC11251

Sitaxsentan sodium; an endothelin A receptor antagonist

Mild to moderate hypertension

Reported preliminary results of Phase II oral safety and tolerance dose-ranging study (10/14)

CENTRAL NERVOUS SYSTEM

Neurobiological Technologies Inc. (OTC BB: NTII) and Merz & Co. GmbH (Germany)

Memantine

Orally administered NMDA receptor antagonist (prevents overactivation of the receptor)

Vascular dementia

Completed two Phase III trials (10/28)

DIABETES

Amylin Pharmaceuticals Inc. (AMLN)

AC2993

Synthetic exendin-4; 39-amino-acid peptide that exhibits anti-diabetic activity similar to the mammalian hormone glucagon-like peptide-1

Type 2 diabetes

Reported results from Phase II trial (10/28)

INFECTION

Cel-Sci Corp. (AMEX:HIV)

Multikine

Natural mixture of human cytokines, including interleukin-2

HIV infection

The company reported that independent investigators completed a clinical study of Multikine to determine safety and its ability to improve immune function (10/19)

ID Biomedical Corp. (Canada; IDBE; TSE:IDB) and the National Institute of Allergy and Infectious Diseases

GAS vaccine

Group A streptococcus vaccine; a subunit vaccine made from the terminal fragments of the surface M protein

Group A streptococcus

Commenced Phase I trial (10/6)

Procept Inc. (PRCT)

PRO 2000 Gel

Microbicide designed to provide protection against HIV infection and other sexually transmitted diseases

HIV and other infections

Initiated clinical safety trial (10/13)

Triangle Pharmaceuticals Inc. (VIRS)

Coactinon

Emivirine; non-nucleoside reverse transcriptase inhibitor

Advanced HIV infection

Modified clinical trial whereby patients will be offered the opportunity to stay on Coactinon with or without nelfinavir, or to change to a regimen that does not include Coactinon (10/7)

Coactinon

Emivirine; non-nucleoside reverse transcriptase inhibitor

Treatment-naive HIV-infected patients

Presented 24-week data from its MKC 301 study at the 7th European Conference on Clinical Aspects and Treatments of HIV Infection in Portugal (10/26)

Trimeris Inc. (TRMS) and Hoffmann-La Roche Inc.(the U.S. subsidiary of F. Hoffmann-La Roche; Switzerland)

T-20

Antiretroviral, fusion inhibitor peptide

HIV infection

Presented 16-week results of Phase II trial at the 7th European Conference on Clinical Aspects and Treatments of HIV Infection in Portugal (10/25)

U.S. Bioscience (AMEX:UBS)

Lodenosine (FddA)

A nucleoside reverse transcriptase inhibitor

HIV infection

Suspended Phase II trial due to serious adverse events, including a patient death (10/14)

VaxGen Inc. (VXGN)

AIDSVax

Vaccine designed to prevent HIV infection; further details ND

HIV infection

Completed patient enrollment and innoculation in U.S. portion of clinical trial (10/12)

MISCELLANEOUS

Abgenix Inc. (ABGX)

ABX-IL8

Fully human monoclonal antibody targeting interleukin-8

Psoriasis

Completed Phase I/II trial (10/5)

Alza Corp. (NYSE:AZA) and Crescendo Pharmaceuticals Corp. (CNDO)

Concerta (Oros methylphenidate)

Methylphenidate HC1 extended release tablets

Attention deficit disorder and attention deficit hyperactivity disorder

Presented clinical study results at the 46th annual meeting of the American Academy of Child and Adolescent Psychiatry in Chicago (10/25)

AnorMed Inc. (Canada; TSE: AOM) and Shire Pharmaceuticals Group plc (UK)

Lambda

A formulation of lanthanum carbonate that binds with dietary phosphate, preventing its absorption in the bloostream

High blood phosphate levels in patients with chronic kidney failure

Commenced Phase III clinical trials in the U.S. (10/19)

Biogen Inc. (BGEN)

Antova

Humanized anti-CD40 ligand monoconal antibody, an immunomodulator that selectively binds to CD40 ligand, a co-stimulatory molecule found on activated T cells

Factor VIII inhibitor syndrome, islet cell transplantation, multiple sclerosis, kidney transplantation, systemic lupus erythematosus, and immune thrombocytopenic purpura

Suspended clinical trials due to adverse incidents involving thrombo-embolic events (10/21)

Celgene Corp. (CELG)

Attendade

D-methylphenidate; chirally pure version of dI-methylphenidate (Ritalin)

Attention deficit disorder and attention deficit hyperactivity disorder

Presented efficacy trial data at the 46th annual meeting of the American Academy of Child and Adolescent Psychiatry in Chicago (10/25)

Corixa Corp. (CRXA) and Allergy Therapeutics Ltd.* (UK)

MPL adjuvant

Immunomodulator for use with allergy desensitization products

Various allergic diseases

Presented data on clinical studies combining MPL with Allergy Therapeutics's Pollinex Quattro allergy vaccines at the Allergie 2000 Symposium at the DGAI conference in Germany (10/27)

Dura Pharmaceuticals (DURA) and Spiros Development Corp. II Inc. (SDCOZ)

Budesonide

Antiasthmatic therapeutic

Asthma

Initiated patient screening for a clinical study designed to establish target dosages by comparing budesonide delivered in the Spiros pulmonary drug delivery system to a commercially available dry powder inhaler form of budesonide (10/26)

Idec Pharmaceuticals (IDPH)

Idec-114

Anti-B7-1 monoclonal antibody that blocks the binding of the CD80 ligand on antigen-presenting cells to the CD28 receptor on T cells, thereby interfering with T-cell activation

Psoriasis

Commenced Phase I/II trial (10/4)

Immunex Corp. (IMNX)

Nuvance

A recombinant human version of a naturally occurring protein thought to act by binding to interleukin-4, a protein present in asthmatic lungs

Asthma

Presented results of Phase I/II trial at the European Respiratory Society meetng in Spain (10/12)

InKine Pharmaceutical Co. Inc. (INKP)

Diacol

Sodium phosphate tablets

Patients undergoing colonoscopies and other procedures

Presented Phase II results at the 1999 Annual Meeting of the American College of Gastroenterology in Arizona (10/12)

Neurocrine Biosciences Inc. (NBIX)

NBI-34060

Non-benzodiazepine compound that binds to specific sites on GABAA receptors

Insomnia

Reported results of clinical comparison studies of NBI-34060 against zaleplon and zolpidem at the Society of Neuroscience conference (10/27)

SkyePharma plc (UK; LSE:SKP) and Novartis Pharma AG (Switzerland)

Foradil

Formoterol fumarate; a fast-onset beta-agonist bronchodilator

Asthma

Commenced clinical trials using Foradil with SkyePharma's multi-dose dry powder inhaler drug delivery technology (10/13)

Peptide Therapeutics Group plc (UK; LSE:PTE)

Arilvax

Single-dose vaccine; further details ND

Yellow fever

Commenced Phase III trials in the U.S. (10/18)

Protein Design Labs Inc. (PDLI)

Humanized anti-CD3 antibody, thought to act by targeting the CD3 antigen on T lymphocytes, a cell type involved in graft rejection

Prevention of acute rejection episodes in kidney transplantation

Initiated a Phase II trial (10/20)

Notes:

* Indicates a privately held company

** The dates listed indicate the issue dates of press releases, and are not necessarily the dates on which stated events took place.

Unless otherwise noted, the stock symbols listed for public companies are on the Nasdaq market.

AMEX = American Stock Exchange; LSE = London Stock Exchange; NYSE = New York Stock Exchange; OTC BB: = Over the Counter Bulletin Board; SSE - Swedish Stock Exchange; TSE = Toronto Stock Exchange

ND = Not disclosed